WIN 56,098

WIN 56,098
Identifiers
	IUPAC name Anthracen-9-yl-{2-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-indol-3-yl}methanone;
CAS Number	134959-50-5;
PubChem CID	9803721;
ChemSpider	7979481;
ChEMBL	ChEMBL105605;
CompTox Dashboard (EPA)	DTXSID801029724 ;
Chemical and physical data
Formula	C30H28N2O2
Molar mass	448.566 g·mol−1
3D model (JSmol)	Interactive image;
	SMILES O=C(c3c1ccccc1cc2ccccc23)c4c6ccccc6n(c4C)CCN5CCOCC5;

WIN 56,098 is a chemical that is considered to be an aminoalkylindole derivative. It is a tricyclic aryl derivative that acts as a competitive antagonist at the CB₂ cannabinoid receptor. Its activity at CB₁ was significantly less effective. WIN 56,098 failed to antagonize any of the in vivo effects of THC.^[1]

References

↑ Howlett AC, Berglund B, Melvin LS (October 1995). "Cannabinoid Receptor Agonists and Antagonists". Current Pharmaceutical Design. 1 (3): 343–352. doi:10.2174/1381612801666220918164118. S2CID 252386978.

[agonistsantagonists-1] Howlett AC, Berglund B, Melvin LS (October 1995). "Cannabinoid Receptor Agonists and Antagonists". Current Pharmaceutical Design. 1 (3): 343–352. doi:10.2174/1381612801666220918164118. S2CID 252386978.

[1]

See also

References